MERCK SHARP & DOHME CORP.
Patent Owner
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- US PATENTS IN FORCE 2,297
- 255 US APPLICATIONS PENDING
- Feb 01, 2018 most recent publication
Details
- 2,297 Issued Patents
- 520 Issued in last 3 years
- 249 Published in last 3 years
- 29,538 Total Citation Count
- Mar 08, 1977 Earliest Filing
- 1,567 Expired/Abandoned/Withdrawn Patents
Patent Activity in the Last 10 Years
20082009201020112012201320142015201620172018
0200400
Technologies
Intl Class
Technology
MATTERS
Rank in Class
Top Patents (by citation)
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Recent Publications
Publication #
Title
Filing Date
Pub Date
Intl Class
2018/0028,509
SUBSTITUTED QUINOLIZINE DERIVATIVES USEFUL AS HIV INTEGRASE INHIBITORS
Oct 05, 17
Feb 01, 18
[C07D, A61K]
2018/0029,981
Process for Making Beta 3 Agonists and Intermediates
Sep 26, 17
Feb 01, 18
[C07D, C12P]
2018/0030,007
ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
Oct 09, 17
Feb 01, 18
[C07D, A61K]
2018/0015,106
PREPARATION AND USE OF 7A-HETEROCYCLE SUBSTITUTED- 6,6-DIFLUORO BICYCLIC HIMBACINE DERIVATIVES AS PAR-1 RECEPTOR ANTAGONISTS
Sep 26, 17
Jan 18, 18
[C07D, A61K]
2018/0016,263
INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL
Feb 08, 16
Jan 18, 18
[C07D, A61K]
2018/0009,807
INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL
Jan 25, 16
Jan 11, 18
[C07D, A61K]
2018/0009,828
IMIDAZOPYRAZINE ANALOGS WITH 3-TERTIARY CARBON SUBSTITUTIONS AS BTK INHIBITORS
Dec 17, 15
Jan 11, 18
[C07D, A61K]
Recent Patents
Patent #
Title
Filing Date
Issue Date
Intl Class
9877957
Tetrahydroisoquinoline derivatives useful as inhibitors of diacylglyceride O-acyltransferase 2
Aug 31, 15
Jan 30, 18
[C07D, C07C, A61K]
9873707
Methods and intermediates for preparing macrolactams
Oct 14, 14
Jan 23, 18
[C07D, C07C, C07K]
9868738
Diazine-fused amidines as BACE inhibitors, compositions, and their use
Sep 14, 15
Jan 16, 18
[C07D]
9861620
Substituted quinolizine derivatives useful as HIV integrase inhibitors
Sep 26, 14
Jan 09, 18
[C07D, A61K]
9861692
Dengue virus vaccine compositions and methods of use thereof
Jun 17, 14
Jan 09, 18
[C12N, A61K, C07K]
9862720
Inhibitors of the renal outer medullary potassium channel
Oct 26, 15
Jan 09, 18
[C07D, A61K]
9862725
Process for preparing chiral dipeptidyl peptidase-IV inhibitors
Jul 16, 15
Jan 09, 18
[C07F, C07D, C07C, A61K]
Expired/Abandoned/Withdrawn Patents
Patent #
Title
Status
Filing Date
Issue/Pub Date
Intl Class
2017/0240,539
Preparation and Use of Cyclic Sulfonamide Derivatives as PAR-1 Receptor Antagonists
ABAN
Oct 09, 15
Aug 24, 17
[C07D]
2017/0166,586
PROCESS FOR MAKING TETRACYCLIC HETEROCYCLE COMPOUNDS
ABAN
Jul 10, 15
Jun 15, 17
[C07F, C07D, C07C]
2016/0311,791
NOVEL TRICYCLIC CALCIUM SENSING RECEPTOR ANTOGONISTS FOR THE TREATMENT OF OSTEOPOSOSIS
ABAN
Dec 17, 14
Oct 27, 16
[C07D, C07C]
2016/0257,697
THIOPHENE-SUBSTITUTED TETRACYCLIC COMPOUNDS AND METHODS OFUSE THEREOF FOR THE TREATMENT OF VIRAL DISEASES
ABAN
Dec 31, 13
Sep 08, 16
[C07D, A61K]
2016/0243,128
POLYCYCLIC HETEROCYCLE DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES
ABAN
May 09, 16
Aug 25, 16
[A61K]
2016/0194,369
METHODS AND COMPOSITIONS FOR CO-EXPRESSION OF POLYPEPTIDES OF INEREST AND IL6
ABAN
Aug 07, 14
Jul 07, 16
[C07K]
2016/0194,660
EXPRESSION VECTORS FOR RECOMBINANT PROTEIN PRODUCTION IN MAMMALIAN CELLS
ABAN
Dec 18, 13
Jul 07, 16
[C12N, C12P, C07K]
2016/0166,529
Formulations for Cathepsin K Inhibitors with Vitamin D
ABAN
Jul 07, 14
Jun 16, 16
[A61K, A61J]
2016/0130,259
SUBSTITUTED BENZOFURAN COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES
ABAN
Jun 19, 14
May 12, 16
[C07D, A61K]
2016/0130,574
METHODS OF MEASURING GENE EXPRESSION IN FACS-SORTED CELLS
ABAN
Apr 02, 14
May 12, 16
[C12N, C12Q, G01N]
2016/0130,659
COMPOSITIONS AND METHODS FOR TREATING CANCER
ABAN
Jun 03, 14
May 12, 16
[C12Q, G01N, C07K]
2016/0114,000
CO-AGONISTS OF THE GLUCAGON AND GLP-1 RECEPTORS
ABAN
Oct 22, 15
Apr 28, 16
[A61K, C07K]
2016/0102,073
2-HYDROXYMETHYL-SUBSTITUTED OREXIN RECEPTOR ANTAGONISTS
ABAN
Apr 21, 14
Apr 14, 16
[C07D]
2016/0084,839
IMMUNOHISTOCHEMICAL ASSAY FOR DETECTING EXPRESSION OF PROGRAMMED DEATH LIGAND 1 (PD-L1) IN TUMOR TISSUE
ABAN
Mar 31, 14
Mar 24, 16
[G01N]
2016/0075,656
QUINOLINE AMIDE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS
ABAN
Nov 18, 15
Mar 17, 16
[C07D]
Top Inventors for This Owner
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