BTK Inhibitors
Number of patents in Portfolio can not be more than 2000
United States of America Patent
Stats
-
Aug 1, 2017
Grant Date -
Jan 12, 2017
app pub date -
Aug 30, 2016
filing date -
Jul 19, 2011
priority date (Note) -
In Force
status (Latency Note)
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Abstract
Provided are 6-5 membered fused pyridine ring compounds according to Formula (I) or pharmaceutically acceptable salts thereof, pharmaceutical compositions comprising these compounds and their use in therapy. In particular, provided is the use of 6-5 membered fused pyridine ring compounds in the treatment of Bruton's Tyrosine Kinase (Btk) mediated disorders.
First Claim
all claims..Other Claims data not available
Family
Country | kind | publication No. | Filing Date | Type | Sub-Type |
---|---|---|---|---|---|
EP | A1 | EP2548877 | Jul 19, 2011 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
APPLICATION PUBLISHED WITH SEARCH REPORT | 4-(5-Membered fused pyridinyl)benzamides as BTK-inhibitors | Jan 23, 2013 | |||
EP | B1 | EP2734529 | Jul 19, 2012 | Patent | Grant |
Type : Patent Sub-Type : Grant | |||||
Patent | BTK INHIBITORS | Sep 05, 2018 | |||
CA | A1 | CA2841899 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
APPLICATION LAID OPEN | BTK INHIBITORS | Jan 24, 2013 | |||
RU | A | RU2014106020 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
LAID OPEN PATENT APPLICATION | ИНГИБИТОРЫ ВТК | Aug 27, 2015 | |||
US | A1 | US20140221333 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
FIRST PUBLISHED PATENT APPLICATION | BTK INHIBITORS | Aug 07, 2014 | |||
BR | A2 | BR112014001279 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
APPLICATION FOR A PATENT OF INVENTION / PIPELINE PATENT PUBLISHED WITHOUT SEARCH REPORT | composto, uso do composto, composição farmacêutica, e, método para tratar um indivíduo que sofre com um distùrbio mediado pela tirosina cinase de bruton (btk) | Jul 24, 2018 | |||
AU | A1 | AU2012286426 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
OPEN TO PUBLIC INSPECTION | BTK inhibitors | Jan 30, 2014 | |||
MX | A | MX2014000747 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
PATENT APPLICATION | INHIBIDORES DE TIROSINA CINASA DE BRUTON. | Oct 15, 2014 | |||
CN | A | CN103917545 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
UNEXAMINED APPLICATION FOR A PATENT FOR INV. | BTK inhibitors | Jul 09, 2014 | |||
JP | A | JP2014520866 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
Published unexamined patent application | BTK INHIBITORS | Aug 25, 2014 | |||
KR | A | KR20140068020 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
UNEXAMINED PATENT APPLICATION | BTK INHIBITORS | Jun 05, 2014 | |||
WO | A1 | WO2013010380 | Jul 19, 2012 | Patent | Application |
Type : Patent Sub-Type : Application | |||||
INTERNATIONAL APPLICATION PUBLISHED WITH INTERNATIONAL SEARCH REPORT | BTK INHIBITORS | Jan 24, 2013 |
- 15 United States
- 10 France
- 8 Japan
- 7 China
- 5 Korea
- 2 Other
Patent Owner(s)
Patent Owner | Address | |
---|---|---|
MERCK SHARP & DOHME LLC | 126 EAST LINCOLN AVE P O BOX 2000 RAHWAY NJ 07065 |
International Classification(s)

- 2016 Application Filing Year
- A61K Class
- 19101 Applications Filed
- 13019 Patents Issued To-Date
- 68.16 % Issued To-Date
Inventor(s)
Inventor Name | Address | # of filed Patents | Total Citations |
---|---|---|---|
Alhassan, Abdul-Basit | Scotch Plains, US | 8 | 51 |
# of filed Patents : 8 Total Citations : 51 | |||
Anand, Rajan | Fanwood, US | 31 | 206 |
# of filed Patents : 31 Total Citations : 206 | |||
Barf, Tjeerd A | Ravenstein, NL | 10 | 72 |
# of filed Patents : 10 Total Citations : 72 | |||
Boga, Sobhana Babu | Scotch Plains, US | 27 | 109 |
# of filed Patents : 27 Total Citations : 109 | |||
Cooper, Alan B | West Caldwell, US | 46 | 365 |
# of filed Patents : 46 Total Citations : 365 | |||
De, Man Adrianus Petrus Antonius | Hurwenen, NL | 22 | 69 |
# of filed Patents : 22 Total Citations : 69 | |||
Gao, Xiaolei | Bridgewater, US | 26 | 134 |
# of filed Patents : 26 Total Citations : 134 | |||
Jans, Christiaan Gerardus Johannes Maria | Cuijk, NL | 22 | 124 |
# of filed Patents : 22 Total Citations : 124 | |||
Kaptein, Allard | Zaltbommel, NL | 42 | 150 |
# of filed Patents : 42 Total Citations : 150 | |||
Kim, Ronald M | Summit, US | 36 | 392 |
# of filed Patents : 36 Total Citations : 392 | |||
Liu, Jian | Edison, US | 667 | 5710 |
# of filed Patents : 667 Total Citations : 5710 | |||
Liu, Shilan | Shanghai, CN | 22 | 110 |
# of filed Patents : 22 Total Citations : 110 | |||
Oubrie, Arthur A | Wijchen, NL | 9 | 54 |
# of filed Patents : 9 Total Citations : 54 | |||
Raaijmakers, Hans C A | Eindhoven, NL | 5 | 40 |
# of filed Patents : 5 Total Citations : 40 | |||
Rewinkel, Johannes Bernardus Maria | Berghem, NL | 24 | 138 |
# of filed Patents : 24 Total Citations : 138 | |||
Sterrenburg, Jan-Gerard | Renkum, NL | 6 | 57 |
# of filed Patents : 6 Total Citations : 57 | |||
Vaccaro, Henry M | South Plainfield, US | 9 | 166 |
# of filed Patents : 9 Total Citations : 166 | |||
Wang, James | Westfield, US | 245 | 6514 |
# of filed Patents : 245 Total Citations : 6514 | |||
Wijkmans, Jacobus C H M | Oss, NL | 6 | 44 |
# of filed Patents : 6 Total Citations : 44 | |||
Wu, Hao | Shanghai, CN | 930 | 3100 |
# of filed Patents : 930 Total Citations : 3100 | |||
Yang, Chundao | Shanghai, CN | 24 | 71 |
# of filed Patents : 24 Total Citations : 71 | |||
Yao, Xin | Westfield, US | 83 | 278 |
# of filed Patents : 83 Total Citations : 278 | |||
Yu, Younong | East Brunswick, US | 57 | 593 |
# of filed Patents : 57 Total Citations : 593 | |||
Zhu, Hugh Y | Warren, US | 14 | 117 |
# of filed Patents : 14 Total Citations : 117 |
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Patent Citation Ranking
- 6 Citation Count
- A61K Class
- 45.09 % this patent is cited more than
- 8 Age
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