Octapeptide compounds derived from somatostatin and the therapeutic use thereof

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United States of America Patent

PATENT NO 9382306
APP PUB NO 20110178013A1
SERIAL NO

13121928

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ATTORNEY / AGENT: (SPONSORED)

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Abstract

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The present invention relates to novel octapeptide compounds of general formula (I): H-2-Nal 1-cyclo(Cys2-Tyr3-AA4-Lys5-Val6-Cys7)-Thr8-NH2. Since these products have a good affinity for certain somatostatin receptor subtypes, they are particularly advantageous for treating pathological states or diseases in which one (or more) somatostatin receptor(s) is (are) involved. These compounds furthermore have physiochemical properties that make it possible to envisage them in diverse solutions for the formulation of medicaments, for example as a pharmaceutically acceptable carrier. The invention also relates to pharmaceutical compositions containing said products and to the use thereof for the preparation of a medicament.

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Patent Owner(s)

Patent OwnerAddress
IPSEN PHARMA S A S65 QUAI GEORGES GORSE BOULOGNE-BILLANCOURT 92100
LE CENTRE NATIONAL DE RECHERCHE SCIENTIFIQUE (CNRS)3 RUE MICHEL-ANGE PARIS F-75794
COMMISSARIAT A LENERGIE ATOMIQUE (CEA)BATIMENT D LE PONNANT 25 RUE LEBLANC PARIS F-75015

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Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Artzner, Franck Cesson Sevigne, FR 4 1
Cherif-Cheikh, Roland Castelldefels, ES 49 422
Cintrat, Jean-Christophe Igny, FR 14 15
Ijsselstijn, Maarten Groningen, NL 1 10
Paternostre, Marie-Thérèse Verrières le Buisson, FR 2 11
Rousseau, Bernard Levallois Perret, FR 6 25
Roux, Stéphane Nice, FR 18 41
Valery, Céline Barelone, ES 2 11

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