Macrocyclic cysteine protease inhibitors and compositions thereof
Number of patents in Portfolio can not be more than 2000
United States of America Patent
Stats
-
Apr 29, 2014
Grant Date -
Jan 27, 2011
app pub date -
Oct 18, 2007
filing date -
Oct 18, 2006
priority date (Note) -
In Force
status (Latency Note)
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Abstract
The present invention provides a novel class of macrocyclic compounds, which are useful as cysteine protease inhibitors. Also provided are novel intermediates and methods of preparing the compounds. The invention also provides pharmaceutical compositions comprising the compounds. The compounds and compositions are useful in methods of treating or preventing one or more diseases associated with cysteine protease activity, particularly those associated with calpain activity.
First Claim
all claims..Other Claims data not available
Family

- 15 United States
- 10 France
- 8 Japan
- 7 China
- 5 Korea
- 2 Other
Patent Owner(s)
Patent Owner | Address | |
---|---|---|
UNIVERSITY OF CANTERBURY | 20 KIRKWOOD AVENUE UPPER RICCARTON CHRISTCHURCH 8041 NEW ZEALAND | |
LINCOLN UNIVERSITY | LINCOLN 7647 | |
DOUGLAS PHARMACEUTICALS LIMITED | LINCOLN AUCKLAND 0610 |
International Classification(s)

- 2007 Application Filing Year
- A61K Class
- 9805 Applications Filed
- 5595 Patents Issued To-Date
- 57.07 % Issued To-Date
Inventor(s)
Inventor Name | Address | # of filed Patents | Total Citations |
---|---|---|---|
Abell, Andrew David | Christchurch, NZ | 4 | 15 |
# of filed Patents : 4 Total Citations : 15 | |||
Aitken, Steven Geoffrey | Christchurch, NZ | 6 | 19 |
# of filed Patents : 6 Total Citations : 19 | |||
Bickerstaffe, Roy | Canterbury, NZ | 3 | 13 |
# of filed Patents : 3 Total Citations : 13 | |||
Coxon, James Morriss | Christchurch, NZ | 3 | 13 |
# of filed Patents : 3 Total Citations : 13 | |||
Duncan, Joanna Kimberley | Christchurch, NZ | 2 | 13 |
# of filed Patents : 2 Total Citations : 13 | |||
Jones, Matthew Alan | Christchurch, NZ | 5 | 13 |
# of filed Patents : 5 Total Citations : 13 | |||
Klanchantra, Mutita | Christchurch, NZ | 2 | 13 |
# of filed Patents : 2 Total Citations : 13 | |||
Lee, Hannah Yun Young | Christchurch, NZ | 2 | 13 |
# of filed Patents : 2 Total Citations : 13 | |||
McNabb, Stephen Brian | Christchurch, NZ | 2 | 13 |
# of filed Patents : 2 Total Citations : 13 | |||
Morton, James David | Canterbury, NZ | 3 | 13 |
# of filed Patents : 3 Total Citations : 13 | |||
Muir, Matthew Stewart | Canterbury, NZ | 3 | 13 |
# of filed Patents : 3 Total Citations : 13 | |||
Neffe, Axel Thomas | Christchurch, NZ | 6 | 15 |
# of filed Patents : 6 Total Citations : 15 | |||
Nikkel, Janna Marie | Christchurch, NZ | 3 | 13 |
# of filed Patents : 3 Total Citations : 13 | |||
Robertson, Lucinda Jane Goodricke | Canterbury, NZ | 2 | 13 |
# of filed Patents : 2 Total Citations : 13 | |||
Stuart, Blair Gibb | Christchurch, NZ | 3 | 13 |
# of filed Patents : 3 Total Citations : 13 |
Cited Art Landscape
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Patent Citation Ranking
- 0 Citation Count
- A61K Class
- 0 % this patent is cited more than
- 11 Age
Forward Cite Landscape
- No Forward Cites to Display

Maintenance Fees
Fee | Large entity fee | small entity fee | micro entity fee | due date |
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11.5 Year Payment | $7400.00 | $3700.00 | $1850.00 | Oct 29, 2025 |
Fee | Large entity fee | small entity fee | micro entity fee |
---|---|---|---|
Surcharge - 11.5 year - Late payment within 6 months | $160.00 | $80.00 | $40.00 |
Surcharge after expiration - Late payment is unavoidable | $700.00 | $350.00 | $175.00 |
Surcharge after expiration - Late payment is unintentional | $1,640.00 | $820.00 | $410.00 |
Full Text

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Mar 30, 2017 | FPAY | FEE PAYMENT | year of fee payment: 4 |
Oct 08, 2013 | I | Issuance | |
Sep 18, 2013 | STCF | INFORMATION ON STATUS: PATENT GRANT | free format text: PATENTED CASE |
Mar 08, 2012 | P | Published | |
Nov 25, 2011 | AS | ASSIGNMENT | free format text: ASSIGNMENT OF ASSIGNORS INTEREST;ASSIGNORS:MIES, STEPHAN;MATTHES, MICHAEL;BOEHNLEIN, JUERGEN;AND OTHERS;SIGNING DATES FROM 20111018 TO 20111025;REEL/FRAME:027314/0578 Owner name: KORSCH AG, GERMANY |
May 06, 2010 | F | Filing | |
May 07, 2009 | PD | Priority Date |

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