2-(2-oxoindoline-3-ylidene)methyl-5-(2-hydroxy-3-morpholin-4-yl-propyl)-6,7-dihydro-1H-pyrrol[3,2-C]pyridine-4(5H)-one compounds and use as protein kinase inhibitors

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United States of America Patent

PATENT NO 8299069
APP PUB NO 20100160317A1
SERIAL NO

12733193

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Abstract

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Pyrrolo[3,2-c]pyridine-4-one-2-indolinone compounds, especially 2-(2-oxoindoline-3-ylidene)methyl-5-(2-hydroxy-3-morpholin-4-yl-propyl)-6,7-dihydro-1H-pyrrol[3,2-c]pyridine-4(5H)-one compounds. Their preparation and pharmaceutical composition, and pharmaceutical use as protein kinase inhibitors.

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Patent Owner(s)

Patent OwnerAddress
SHANGHAI HENGRUI PHARMACEUTICAL CO LTDNO 279 WENJING ROAD MINHANG DISTRICT SHANGHAI 200245
JIANGSU HENGRUI MEDICINE CO LTD222047 NO 7 KUNLUN MOUNTAIN ROAD LIANYUNGANG ECONOMIC AND TECHNOLOGICAL DEVELOPMENT ZONE JIANGSU LIANYUNGANG CITY JIANGSU PROVINCE 222047

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Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Su, Yidong Shanghai, CN 17 143
Tang, Peng Cho Shanghai, CN 162 3817
Yang, Jialiang Shanghai, CN 7 33
Zhao, Fuqiang Shanghai, CN 19 88

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