2-[1H-benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides as kinase inhibitors

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United States of America Patent

PATENT NO 8129396
APP PUB NO 20100081653A1
SERIAL NO

12567060

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2-[1H-benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and their salts are kinase inhibitors, useful in the treatment of cancer.

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TELIK INC750-H GATEWAY BOULEVARD SAN FRANCISCO CA 94080

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Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Aurrecoechea, Natalia Oakland, US 12 30
Beroza, Paul P Belmont, US 5 42
Damodaran, Komath V Cupertino, US 3 0
Pontius, Karen Y Aromas, US 1 0
Robinson, Louise San Carlos, US 14 92
Simon, Reyna J Los Gatos, US 25 267
Vu, Truong San Martin, US 1 0
Weber, Kevin T Carmel, US 10 48

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