Peptidyl sulfonyl imidazolides as selective inhibitors of serine proteases
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United States of America Patent
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Mar 19, 2002
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app pub date -
Nov 22, 1999
filing date -
Nov 22, 1999
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Abstract
Novel .alpha.-amino and peptidyl sulfonyl imidazolides, a method for their synthesis, and a method for inhibiting serine proteases therewith are disclosed. Pharmaceutical compositions containing .alpha.-amino and peptidyl sulfonyl imidazolides and their use in the treatment of disease states characterized by an over-activity of serine proteases are also disclosed. Novel synthetic methods for the synthesis of sulfonyl derivatives, particularly .alpha.-amino and peptidyl sulfonyl derivatives, from thioic acid S-esters are also disclosed.
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