BIFUNCTIONAL PROTAC-TYPE COMPOUNDS TARGETING PXR, METHOD FOR PREPARING SAME AND THERAPEUTIC USE THEREOF

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United States of America Patent

APP PUB NO 20240252658A1
SERIAL NO

18562251

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Abstract

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The present application relates to novel bifunctional PROTAC-type compounds simultaneously binding the target protein PXR and E3-ubiquitin ligase, to a method for preparing same, and to uses thereof for treating cancers overexpressing PXR.

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Patent Owner(s)

Patent OwnerAddress
CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE3 RUE MICHEL ANGE PARIS 75016
INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE101 RUE DE TOLBIAC PARIS 75013
UNIVERSITÉ DE MONTPELLIER163 RUE AUGUSTE BROUSSONNET MONTPELLIER 34090
ECOLE NATIONALE SUPERIEURE DE CHIMIE DE MONTPELLIER240 AVENUE DU PROFESSEUR EMILE JEANBRAU MONTPELLIER CEDEX 5 34296

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Inventor(s)

Inventor Name Address # of filed Patents Total Citations
AMBLARD-CAUSSIL, Muriel SAINT VINCENT DE BARBEYRARGUES, FR 5 0
BOURGUET, William SAINT GELY DU FESC, FR 2 0
CHAVANIEU, Alain ASSAS, FR 2 89
DELFOSSE, Vanessa PRADES-LE-LEZ, FR 1 0
GERBAL-CHALOIN, Sabine PRADES-LE-LEZ, FR 1 0
LACONDE, Guillaume MONTPELLIER, FR 3 0
PANNEQUIN, Julie SÈTE, FR 10 32
PASCUSSI, Jean-Marc VERGEZE, FR 1 0

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