PROCESS FOR THE PREPARATION OF 3ALPHA-HYDROXY-5ALPHA-PREGNAN-20-0NE (BREXANOLONE)

Number of patents in Portfolio can not be more than 2000

United States of America

APP PUB NO 20210388020A1
SERIAL NO

17282772

Stats

ATTORNEY / AGENT: (SPONSORED)

Importance

Loading Importance Indicators... loading....

Abstract

See full text

The present invention relates to a new process for the synthesis of 3α-hydroxy-5α-pregnan-20-one, commonly known as brexanolone, wherein the corresponding cyclic 20-ketal or cyclic 20-thioketal compound of formula (IV) is deprotected with the use or iodine in an organic solvent: (I).

Loading the Abstract Image... loading....

First Claim

See full text

Family

Loading Family data... loading....

Patent Owner(s)

Patent OwnerAddress
INDUSTRIALE CHIMICA S R LVIA ABBONDIO SANGIORGIO 12 MILAN 20145

International Classification(s)

  • [Classification Symbol]
  • [Patents Count]

Inventor(s)

Inventor Name Address # of filed Patents Total Citations
BORELLI, Tea COMO, IT 1 0
DELFRATE, Claudio RHO, IT 4 0
LENNA, Roberto S. GIORGIO SU LEGNANO, IT 29 20
RIGAMONTI, Davide ERBA, IT 3 0

Cited Art Landscape

Load Citation

Patent Citation Ranking

Forward Cite Landscape

Load Citation