1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-ones and 1,5-dihydro-4H-pyrazolo[4,3-c]pyridin-4-ones as PDE1 Inhibitors

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United States of America Patent

APP PUB NO 20170291901A1
SERIAL NO

15481083

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Abstract

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The present invention provides 1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-ones and 1,5-dihydro-4H-pyrazolo[4,3-c]pyridin-4-ones of formula (I) as PDE1 inhibitors and their use as a medicament, in particular for the treatment of neurodegenerative disorders and psychiatric disorders.

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Patent Owner(s)

Patent OwnerAddress
H LUNDBECK A/S2500 VALBY

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Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Jessing, Mikkel Valby, DK 40 291
Juhl, Karsten Valby, DK 68 444
Kehler, Jan Valby, DK 79 392
Langgård, Morten Valby, DK 46 279
Marigo, Mauro Valby, DK 55 305
Rasmussen, Lars Kyhn Valby, DK 53 337
Vital, Paulo Jorge Vieira Valby, DK 25 231

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