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Country	kind	publication No.	Filing Date	Type	Sub-Type
TW	A	TW201311698	Aug 10, 2012	Patent	Application
Type : Patent Sub-Type : Application
LAID OPEN APPLICATION FOR PATENT OR PATENT OF ADDITION		1,4-diazabicyclo[3.2.2]nonanes as neuronal nicotinic acetylcholine receptor ligands		Mar 16, 2013
JP	A	JP2014524470	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
Published unexamined patent application		1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS		Sep 22, 2014
EP	A1	EP2748170	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
APPLICATION PUBLISHED WITH SEARCH REPORT		1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS		Jul 02, 2014
MX	A	MX2014002005	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
PATENT APPLICATION		1,4-DIAZABICICLO[3.2.2]NONANOS COMO LIGANDOS DE RECEPTORES NICOTINICOS NEURONALES DE ACETILCOLINA.		Mar 27, 2014
WO	A1	WO2013028587	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
INTERNATIONAL APPLICATION PUBLISHED WITH INTERNATIONAL SEARCH REPORT		1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS		Feb 28, 2013
AU	A1	AU2012299077	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
OPEN TO PUBLIC INSPECTION		1,4-diazabicyclo(3.2.2)nonanes as neuronal nicotinic acetylcholine receptor ligands		Mar 13, 2014
CN	A	CN103797016	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
UNEXAMINED APPLICATION FOR A PATENT FOR INV.		1,4-diazabicyclo[3.2.2]nonanes as neuronal nicotinic acetylcholine receptor ligands		May 14, 2014
CA	A1	CA2844764	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
APPLICATION LAID OPEN		1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS		Feb 28, 2013
RU	A	RU2014110971	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
LAID OPEN PATENT APPLICATION		1,4-ДИАЗАБИЦИКЛО[3.2.2]НОНАНЫ В КАЧЕСТВЕ ЛИГАНДОВ ДЛЯ НЕЙРОННЫХ НИКОТИНОВЫХ АЦЕТИЛХОЛИНОВЫХ РЕЦЕПТОРОВ		Sep 27, 2015
BR	A2	BR112014004068	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
APPLICATION FOR A PATENT OF INVENTION / PIPELINE PATENT PUBLISHED WITHOUT SEARCH REPORT		1,4-diazabiciclo [3.2.2] nonanos como ligantes do receptor acetilcolina nicotínico neuronal		Mar 14, 2017
PH	A1	PH12014500413	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
Patent Application		1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS		Apr 14, 2014
KR	A	KR20140068079	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
UNEXAMINED PATENT APPLICATION		1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS		Jun 05, 2014
SG	A	SG2014011126	Aug 20, 2012	Patent	Grant
Type : Patent Sub-Type : Grant
UK PATENTS REGISTERED		1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS		Jun 27, 2014
PE	A1	PE20141247	Aug 20, 2012	Patent	Application
Type : Patent Sub-Type : Application
PATENT APPLICATION		1,4-DIAZABICICLO[3.2.2]NONANOS COMO LIGANDOS DE RECEPTORES NICOTINICOS NEURONALES DE ACETILCOLINA		Oct 12, 2014
AR	A1	AR087602	Aug 21, 2012	Patent	Application
Type : Patent Sub-Type : Application
INDEPENDENT PATENT APPLICATION		1,4-DIAZABICICLO[3.2.2]NONANOS COMO LIGANDOS DE RECEPTORES NICOTINICOS NEURONALES DE ACETILCOLINA		Apr 03, 2014
UY	A	UY34281	Aug 21, 2012	Patent	Application
Type : Patent Sub-Type : Application
PATENT APPLICATION		'1,4-DIAZABICICLO[3.2.2]NONANOS COMO LIGANDOS DE RECEPTORES NICOTÍNICOS NEURONALES DE ACETILCOLINA		Feb 28, 2014
IL	A0	IL230889	Feb 09, 2014	Patent	Application
Type : Patent Sub-Type : Application
PATENT APPLICATION FILED		1,4-diazabicyclo[3.2.2]nonanes as neuronal nicotinic acetylcholine receptor ligands		Jan 01, 1970
CL	A1	CL2014000417	Feb 20, 2014	Patent	Application
Type : Patent Sub-Type : Application
PATENT APPLICATION		Compuestos derivados de 1,4-diazabiciclo[3.2.2]nonanos, como ligandos de receptores nicotinicos neuronales de acetilcolina; composicion farmaceutica que los comprende; y su uso para el tratamiento de enfermedades inflamatorias y enfermedades asociadas a la disfuncion del sistema nervioso central.		Sep 26, 2014
CO	A2	CO6920290	Mar 20, 2014	Patent	Application
Type : Patent Sub-Type : Application
APPLICATION DERIVED FROM A PCT APPLICATION		1,4-diazabiciclo[3.2.2]nonanos como ligandos de receptores nicotínicos neuronales de acetilcolina		Apr 10, 2014

• 15 United States
• 10 France
• 8 Japan
• 7 China
• 5 Korea
• 2 Other

Patent Owner(s)

Patent Owner	Address
TARGACEPT INC	WINSTON-SALEM NC

International Classification(s)

• A61K:PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOS....
• C07D:HETEROCYCLIC COMPOUNDS

Inventor(s)

Inventor Name	Address	# of filed Patents	Total Citations
Mazurov, Anatoly	Greensboro, US	24	59
# of filed Patents : 24 Total Citations : 59
Miao, Lan	Advance, US	35	215
# of filed Patents : 35 Total Citations : 215
Showalter, Todd	Clemmons, US	11	8
# of filed Patents : 11 Total Citations : 8

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Patent Citation Ranking

• 1 Citation Count
• A61K Class

• 21.20 % this patent is cited more than
• 11 Age

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Maintenance Fees

Fee	Large entity fee	small entity fee	micro entity fee	due date
11.5 Year Payment	$7400.00	$3700.00	$1850.00	Mar 4, 2026

Fee	Large entity fee	small entity fee	micro entity fee
Surcharge - 11.5 year - Late payment within 6 months	$160.00	$80.00	$40.00
Surcharge after expiration - Late payment is unavoidable	$700.00	$350.00	$175.00
Surcharge after expiration - Late payment is unintentional	$1,640.00	$820.00	$410.00

Full Text

US Patent Application No: 2014/0249,141

1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS

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Abstract

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The present invention relates to compounds that bind to and modulate the activity of neuronal nicotinic acetylcholine receptors, to processes for preparing these compounds, to pharmaceutical compositions containing these compounds, and to methods of using these compounds for treating a wide variety of conditions and disorders, including inflammatory diseases and diseases associated with dysfunction of the central nervous system (CNS).

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Description

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Claims

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