A3 adenosine receptor allosteric modulators
Number of patents in Portfolio can not be more than 2000
United States of America Patent
Stats
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May 3, 2016
Grant Date -
Aug 1, 2013
app pub date -
Mar 13, 2013
filing date -
Jan 26, 2006
priority date (Note) -
In Force
status (Latency Note)
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Abstract
The claimed subject matter relates to allosteric modulation of A3 adenosine receptor (A3AR) and provides for the use of an A3 adenosine receptor modulator (A3RM), for the preparation of pharmaceutical compositions for modulating the A3AR in a subject, as well as pharmaceutical compositions including the same and therapeutic methods including administering to a subject an amount of an A3RM, the amount being effective to modulate A3AR activity. The A3RM according to claimed subject matter are 1H-Imidazo-[4,5-c]quinolin-4-amine derivatives. Also provided are 1H-Imidazo-[4,5-c]quinolin-4-amine derivatives.
First Claim
all claims..Other Claims data not available
Family

- 15 United States
- 10 France
- 8 Japan
- 7 China
- 5 Korea
- 2 Other
Patent Owner(s)
Patent Owner | Address | |
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THE UNITED STATES OF AMERICA REPRESENTED BY THE SECRETARY DEPT OF HEALTH AND HUMAN SERVICES | WASHINGTON DC |
International Classification(s)

- 2013 Application Filing Year
- A61K Class
- 12711 Applications Filed
- 11051 Patents Issued To-Date
- 86.95 % Issued To-Date
Inventor(s)
Inventor Name | Address | # of filed Patents | Total Citations |
---|---|---|---|
Brussee, Johannes | Rijnsburg, NL | 12 | 53 |
# of filed Patents : 12 Total Citations : 53 | |||
Göblyös, Anikó | Ujszasz, HU | 1 | 0 |
# of filed Patents : 1 Total Citations : 0 | |||
Gao, Zhan-Guo | Rockville, US | 2 | 9 |
# of filed Patents : 2 Total Citations : 9 | |||
Ijzerman, Adriaan P | Haarlem, NL | 5 | 32 |
# of filed Patents : 5 Total Citations : 32 | |||
Jacobson, Kenneth | Silver Spring, US | 4 | 84 |
# of filed Patents : 4 Total Citations : 84 |
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Patent Citation Ranking
- 0 Citation Count
- A61K Class
- 0 % this patent is cited more than
- 9 Age
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Maintenance Fees
Fee | Large entity fee | small entity fee | micro entity fee | due date |
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11.5 Year Payment | $7400.00 | $3700.00 | $1850.00 | Nov 3, 2027 |
Fee | Large entity fee | small entity fee | micro entity fee |
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Surcharge - 11.5 year - Late payment within 6 months | $160.00 | $80.00 | $40.00 |
Surcharge after expiration - Late payment is unavoidable | $700.00 | $350.00 | $175.00 |
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