A3 adenosine receptor allosteric modulators

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United States of America Patent

PATENT NO 9326978
APP PUB NO 20130197025A1
SERIAL NO

13800560

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ATTORNEY / AGENT: (SPONSORED)

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Abstract

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The claimed subject matter relates to allosteric modulation of A3 adenosine receptor (A3AR) and provides for the use of an A3 adenosine receptor modulator (A3RM), for the preparation of pharmaceutical compositions for modulating the A3AR in a subject, as well as pharmaceutical compositions including the same and therapeutic methods including administering to a subject an amount of an A3RM, the amount being effective to modulate A3AR activity. The A3RM according to claimed subject matter are 1H-Imidazo-[4,5-c]quinolin-4-amine derivatives. Also provided are 1H-Imidazo-[4,5-c]quinolin-4-amine derivatives.

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Patent Owner(s)

Patent OwnerAddress
THE UNITED STATES OF AMERICA REPRESENTED BY THE SECRETARY DEPT OF HEALTH AND HUMAN SERVICESWASHINGTON DC

International Classification(s)

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  • 2013 Application Filing Year
  • A61K Class
  • 12711 Applications Filed
  • 11051 Patents Issued To-Date
  • 86.95 % Issued To-Date
Click to zoom InYear of Issuance% of Matters IssuedCumulative IssuancesYearly Issuances2013201420152016201720182019202020212022202320240255075100

Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Brussee, Johannes Rijnsburg, NL 12 53
Göblyös, Anikó Ujszasz, HU 1 0
Gao, Zhan-Guo Rockville, US 2 9
Ijzerman, Adriaan P Haarlem, NL 5 32
Jacobson, Kenneth Silver Spring, US 4 84

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  • A61K Class
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Citation count rangeNumber of patents cited in rangeNumber of patents cited in various citation count ranges6209860894426710349291291182201 - 1011 - 2021 - 3031 - 4041 - 5051 - 6061 - 7071 - 8081 - 9091 - 100100 +0500100015002000250030003500400045005000550060006500700075008000850090009500

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11.5 Year Payment $7400.00 $3700.00 $1850.00 Nov 3, 2027