Prodrugs of substituted triazole derivatives and uses thereof

Number of patents in Portfolio can not be more than 2000

United States of America

PATENT NO 11298367
APP PUB NO 20200338096A1
SERIAL NO

16758742

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Abstract

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The present invention relates to prodrugs of 3-({3-(4-chlorophenyl)-5-oxo-4-[(2S)-3,3,3-trifluoro-2-hydroxypropyl ]-4,5-dihydro-1H-1,2,4-triazol-1-yl}methyl)-1-[3-(trifluoromethyl)-pyridin-2-yl ]-1H-1,2,4-triazole-5-carboxamide, 3-({3-(4-chlorophenyl)-5-oxo-4-[(2S)-3,3,3-trifluoro-2-hydroxypropyl ]-4,5-dihydro-1H-1,2,4-triazol-1-yl}methyl)-1-[2-(trifluoromethyl)-phenyl]-1H-1,2,4-triazole-5-carboxamide and 3-({3-(4-chlorophenyl)-5-oxo-4-[(2S)-3,3,3-trifluoro-2-hydroxypropyl ]-4,5-dihydro-1H-1,2,4-triazol-1-yl}methyl)-1-(3-chloropyridin-2-yl)-1H-1,2,4-triazole-5-carboxamide, to processes for the preparation of such compounds, to pharmaceutical compositions containing such compounds, and to the use of such compounds or compositions for the treatment and/or prevention of diseases, in particular for the treatment and/or prevention of renal and cardiovascular diseases.

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Patent Owner(s)

Patent OwnerAddress
BAYER AKTIENGESELLSCHAFT51373 LEVERKUSEN
BAYER PHARMA AKTIENGESELLSCHAFT13353 BERLIN

International Classification(s)

Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Buchmueller, Anja Essen, DE 3 5
Cernecka, Hana Wuppertal, DE 9 38
Collin-Kroepelin, Marie-Pierre Wuppertal, DE 8 5
Droebner, Karoline Velbert, DE 4 5
Fricke, Robert Cologne, DE 2 52
Fuerstner, Chantal Muelheim/Ruhr, DE 21 41
Kolkhof, Peter Wuppertal, DE 65 359
Krenz, Ursula Leichlingen, DE 27 152
Kretschmer, Axel Wuppertal, DE 42 439
Levilain, Guillaume Wuppertal, DE 11 18
Lustig, Klemens Wuppertal, DE 71 458
Mondritzki, Thomas Essen, DE 23 78
Neubauer, Thomas Wuppertal, DE 29 91
Pook, Elisabeth Wuppertal, DE 38 197
Schirmer, Heiko Solingen, DE 59 134
Schmeck, Carsten Muelheim, DE 72 425
Tinel, Hanna Wuppertal, DE 52 196
Wasnaire, Pierre Duesseldorf, DE 82 524
Witowski, Norbert Wolfenbuettel, DE 8 140
Wittwer, Matthias Beat Riehen, CH 23 86

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