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Patent Activity in the Last 10 Years

Technologies

Intl Class Technology Matters Rank in Class
 
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 32223
 
 
 
C07D HETEROCYCLIC COMPOUNDS 29133
 
 
 
C07C ACYCLIC OR CARBOCYCLIC COMPOUNDS 3135
 
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 247
 
 
 
C01C AMMONIA; CYANOGEN; COMPOUNDS THEREOF 113

Top Patents (by citation)

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Recent Publications

Publication # Title Filing Date Pub Date Intl Class
2010/0249,165 PDZ DOMAIN MODULATORSJun 03, 08Sep 30, 10[A61K, C07D, C07C, A61P]

Recent Patents

Patent # Title Filing Date Issue Date Intl Class
7429618 Potassium channel modulatorsMar 07, 07Sep 30, 08[A61K]
6288079 Tropane-derivatives, their preparation and useJul 10, 98Sep 11, 01[A61K, C07D, A61P]
6124285 Indole-2,3-dione-3-oxime derivativesJun 01, 98Sep 26, 00[A61K, C07D]
5998405 Fused tropane-derivatives as neurotransmitter reuptake inhibitorsJun 04, 98Dec 07, 99[A61K, C07D]
5990312 Method for the preparation of esters of anhydroecgonineNov 04, 97Nov 23, 99[C07D]
5981539 Piperidine compounds as calcium channel blockersMay 29, 98Nov 09, 99[A61K, C07D]
5922724 Benzimidazole compounds and their use as modulators of the GABA a receptor complexFeb 05, 98Jul 13, 99[A61K]
5922725 Benzimidazole compounds and their use as modulators of the GABA.sub.A receptor complexDec 23, 97Jul 13, 99[A61K, C07D]
5902813 Benzimidazole compounds, pharmaceutical compositions containing the compounds and their useJan 28, 98May 11, 99[A61K]
5892047 Process for the preparation of substituted 4-ethyl-piperidines and an intermediate for the preparation of sameAug 04, 97Apr 06, 99[A61K, C07D]

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Expired/Abandoned/Withdrawn Patents

Patent # Title Status Filing Date Issue/Pub Date Intl Class
2012/0309,792 TETRAZOLE DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORSAbandonedDec 16, 10Dec 06, 12[A61K, C07D, A61P]
2012/0238,547 2, 3, 6 - TRIAMINO SUBSTITUTED PYRIDINES AS KV7 (KCNQ) CHANNEL MODULATORSAbandonedSep 02, 10Sep 20, 12[A61K, C07D, A61P]
2012/0238,553 NOVEL BENZODIOXOLYL-OXADIAZOLYL-DIAZABICYCLONONANE DERIVATIVES AND THEIR MEDICAL USEAbandonedJan 25, 10Sep 20, 12[A61K, C07D, A61P]
2012/0232,058 SUBSTITUTED PYRIDINE DERIVATIVES AND THEIR MEDICAL USEAbandonedSep 02, 10Sep 13, 12[A61K, C07D, A61P]
2012/0220,604 PIPERAZINYL-ALKYL-BENZOIMIDAZOL-2-ONE DERIVATIVES AND THEIR USE AS MONOAMINE NEUROTRANSMITTER RE-UPTAKE INHIBITORSAbandonedSep 13, 10Aug 30, 12[A61K, C07D, A61P]
2012/0115,900 SUBSTITUTED NAPHTHYRIDINE DERIVATIVES AND THEIR MEDICAL USEAbandonedApr 21, 10May 10, 12[A61K, C07D, A61P]
2012/0095,025 SUBSTITUTED [1,2,4]TRIAZOLO[1,5-a]PYRIMIDINES AND THEIR USE AS POTASSIUM CHANNEL MODULATORSAbandonedMar 30, 10Apr 19, 12[A61K, C07D, A61P]
2012/0095,056 2,5-DISUBSTITUTED TETRAZOLE DERIVATIVES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORSAbandonedMar 17, 10Apr 19, 12[A61K, C07D, A61P]
2012/0071,469 NOVEL 1,4-DIAZA-BICYCLO[3.2.1]OCTANE DERIVATIVES USEFUL AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORSAbandonedMay 12, 10Mar 22, 12[A61K, C07D, A61P]
2012/0071,471 NOVEL BENZOXAZINONE DERIVATIVES USEFUL FOR THE TREATMENT OF CNS DISORDERSAbandonedMar 11, 10Mar 22, 12[A61K, C07D, A61P]
2012/0059,037 SUBSTITUTED PYRIDINE DERIVATIVES AND THEIR MEDICAL USEAbandonedMar 11, 10Mar 08, 12[A61K, C07D, A61P]
8110588 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptorsExpiredAug 06, 08Feb 07, 12[A61K, C07D]
2012/0028,967 NOVEL DIAZA-BICYCLONONYL-PYRIMIDINYL DERIVATIVES AND THEIR MEDICAL USEAbandonedJan 20, 10Feb 02, 12[A61K, C07D, A61P]
2012/0028,968 NOVEL DIBENZOFURANYL-OXADIAZOLYL-DIAZABICYCLONONANE DERIVATIVES AND THEIR MEDICAL USEAbandonedJan 25, 10Feb 02, 12[A61K, C07D, A61P]
2012/0015,977 QUINOLINONE DERIVATIVES USEFUL FOR THE TREATMENT OF CNS DISORDERSAbandonedJan 18, 10Jan 19, 12[A61K, C07D, A61P]
2012/0004,214 N-OXIDES OF 1,4-DIAZA-BICYCLO[3.2.2]NONYL PYRIMIDINYL DERIVATIVES USEFUL AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDSAbandonedJan 20, 10Jan 05, 12[A61K, C07D, A61P]
2012/0004,215 N-OXIDES OF DIAZABICYCLONONYL PYRIMIDINE DERIVATIVES AND THEIR MEDICAL USEAbandonedJan 25, 10Jan 05, 12[A61K, C07D, A61P]
2012/0004,246 PURINYL DERIVATIVES AND THEIR USE AS POTASSIUM CHANNEL MODULATORSAbandonedMar 27, 08Jan 05, 12[A61K, C07D, A61P]
2012/0004,257 NOVEL COMPOUNDSAbandonedJun 30, 11Jan 05, 12[A61K, C07D, A61P]
2011/0319,397 NOVEL N-OXIDES OF FURANYL-OXADIAZOLYL-DIAZABICYCLONONANE DERIVATIVES AND THEIR MEDICAL USEAbandonedJan 25, 10Dec 29, 11[A61K, C07D, A61P]

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