MERCK SHARP & DOHME CORP.

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Patent Activity in the Last 10 Years

Technologies

Intl Class Technology MATTERS Rank in Class
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 1546 4
 
 
C07D HETEROCYCLIC COMPOUNDS 1215 1
 
 
C07K PEPTIDES 246 11
 
 
A01N PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF 176 11
 
 
C12N MICRO-ORGANISMS OR ENZYMES; COMPOSITIONS THEREOF 170 41
 
 
C07H SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS 137 13
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 107 2
 
 
C07C ACYCLIC OR CARBOCYCLIC COMPOUNDS 102 51
 
 
C12P FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE 91 26
 
 
G01N INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES 68 130
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Top Patents (by citation)

Recent Publications

Publication # Title Filing Date Pub Date Intl Class
2018/0028,509 SUBSTITUTED QUINOLIZINE DERIVATIVES USEFUL AS HIV INTEGRASE INHIBITORS Oct 05, 17 Feb 01, 18 [C07D, A61K]
2018/0029,981 Process for Making Beta 3 Agonists and Intermediates Sep 26, 17 Feb 01, 18 [C07D, C12P]
2018/0030,007 ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS Oct 09, 17 Feb 01, 18 [C07D, A61K]
2018/0030,036 Factor IXa Inhibitors Dec 07, 15 Feb 01, 18 [C07D]
2018/0022,747 Factor IXa Inhibitors Feb 12, 16 Jan 25, 18 [C07D]
2018/0015,106 PREPARATION AND USE OF 7A-HETEROCYCLE SUBSTITUTED- 6,6-DIFLUORO BICYCLIC HIMBACINE DERIVATIVES AS PAR-1 RECEPTOR ANTAGONISTS Sep 26, 17 Jan 18, 18 [C07D, A61K]
2018/0016,263 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Feb 08, 16 Jan 18, 18 [C07D, A61K]
2018/0009,796 ISOQUINOLINE DERIVATIVES AS MGAT2 INHIBITORS Jan 20, 15 Jan 11, 18 [C07D]
2018/0009,807 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Jan 25, 16 Jan 11, 18 [C07D, A61K]
2018/0009,828 IMIDAZOPYRAZINE ANALOGS WITH 3-TERTIARY CARBON SUBSTITUTIONS AS BTK INHIBITORS Dec 17, 15 Jan 11, 18 [C07D, A61K]

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Recent Patents

Patent # Title Filing Date Issue Date Intl Class
9877957 Tetrahydroisoquinoline derivatives useful as inhibitors of diacylglyceride O-acyltransferase 2 Aug 31, 15 Jan 30, 18 [C07D, C07C, A61K]
9872906 Ceftolozane antibiotic compositions Sep 16, 15 Jan 23, 18 [A61K]
9872962 Dual chamber mixing syringes and methods of using same Dec 17, 13 Jan 23, 18 [A61M]
9873707 Methods and intermediates for preparing macrolactams Oct 14, 14 Jan 23, 18 [C07D, C07C, C07K]
9868727 Factor XIa inhibitors Jul 23, 15 Jan 16, 18 [C07D, A61K]
9868733 Azabenzimidazole tetrahydrofuran derivatives Aug 19, 13 Jan 16, 18 [C07D, C07C, A61K]
9868738 Diazine-fused amidines as BACE inhibitors, compositions, and their use Sep 14, 15 Jan 16, 18 [C07D]
9868777 CMV neutralizing antigen binding proteins Jun 09, 14 Jan 16, 18 [C12Q, A61K, C07K]
9861620 Substituted quinolizine derivatives useful as HIV integrase inhibitors Sep 26, 14 Jan 09, 18 [C07D, A61K]
9861692 Dengue virus vaccine compositions and methods of use thereof Jun 17, 14 Jan 09, 18 [C12N, A61K, C07K]
9862707 TrkA kinase inhibitors, compositions and methods thereof Mar 23, 15 Jan 09, 18 [C07D]
9862716 TRKA kinase inhibitors, compositions and methods thereof Mar 23, 15 Jan 09, 18 [C07D]
9862720 Inhibitors of the renal outer medullary potassium channel Oct 26, 15 Jan 09, 18 [C07D, A61K]
9862725 Process for preparing chiral dipeptidyl peptidase-IV inhibitors Jul 16, 15 Jan 09, 18 [C07F, C07D, C07C, A61K]

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Expired/Abandoned/Withdrawn Patents

Patent # Title Status Filing Date Issue/Pub Date Intl Class
2017/0240,539 Preparation and Use of Cyclic Sulfonamide Derivatives as PAR-1 Receptor Antagonists ABAN Oct 09, 15 Aug 24, 17 [C07D]
2017/0216,295 CCR9 ANTAGONIST COMPOUNDS ABAN Jul 27, 15 Aug 03, 17 [C07D, A61K]
2017/0166,586 PROCESS FOR MAKING TETRACYCLIC HETEROCYCLE COMPOUNDS ABAN Jul 10, 15 Jun 15, 17 [C07F, C07D, C07C]
2017/0008,906 INHIBITORS OF HEPATITIS C VIRUS REPLICATION ABAN Sep 22, 16 Jan 12, 17 [C07D, A61K]
2016/0311,791 NOVEL TRICYCLIC CALCIUM SENSING RECEPTOR ANTOGONISTS FOR THE TREATMENT OF OSTEOPOSOSIS ABAN Dec 17, 14 Oct 27, 16 [C07D, C07C]
2016/0279,140 CEFTOLOZANE ANTIBIOTIC COMPOSITIONS ABAN Mar 31, 16 Sep 29, 16 [A61K]
2016/0257,697 THIOPHENE-SUBSTITUTED TETRACYCLIC COMPOUNDS AND METHODS OFUSE THEREOF FOR THE TREATMENT OF VIRAL DISEASES ABAN Dec 31, 13 Sep 08, 16 [C07D, A61K]
2016/0243,128 POLYCYCLIC HETEROCYCLE DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES ABAN May 09, 16 Aug 25, 16 [A61K]
2016/0229,839 Factor XIa Inhibitors ABAN Sep 23, 14 Aug 11, 16 [A01N, C07D]
2016/0194,369 METHODS AND COMPOSITIONS FOR CO-EXPRESSION OF POLYPEPTIDES OF INEREST AND IL6 ABAN Aug 07, 14 Jul 07, 16 [C07K]
2016/0194,660 EXPRESSION VECTORS FOR RECOMBINANT PROTEIN PRODUCTION IN MAMMALIAN CELLS ABAN Dec 18, 13 Jul 07, 16 [C12N, C12P, C07K]
2016/0166,529 Formulations for Cathepsin K Inhibitors with Vitamin D ABAN Jul 07, 14 Jun 16, 16 [A61K, A61J]
2016/0130,259 SUBSTITUTED BENZOFURAN COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES ABAN Jun 19, 14 May 12, 16 [C07D, A61K]
2016/0130,574 METHODS OF MEASURING GENE EXPRESSION IN FACS-SORTED CELLS ABAN Apr 02, 14 May 12, 16 [C12N, C12Q, G01N]
2016/0130,659 COMPOSITIONS AND METHODS FOR TREATING CANCER ABAN Jun 03, 14 May 12, 16 [C12Q, G01N, C07K]
2016/0114,000 CO-AGONISTS OF THE GLUCAGON AND GLP-1 RECEPTORS ABAN Oct 22, 15 Apr 28, 16 [A61K, C07K]
2016/0102,073 2-HYDROXYMETHYL-SUBSTITUTED OREXIN RECEPTOR ANTAGONISTS ABAN Apr 21, 14 Apr 14, 16 [C07D]
2016/0084,839 IMMUNOHISTOCHEMICAL ASSAY FOR DETECTING EXPRESSION OF PROGRAMMED DEATH LIGAND 1 (PD-L1) IN TUMOR TISSUE ABAN Mar 31, 14 Mar 24, 16 [G01N]
2016/0075,645 AMIDATION PROCESS ABAN Nov 23, 15 Mar 17, 16 [C07C]
2016/0075,656 QUINOLINE AMIDE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS ABAN Nov 18, 15 Mar 17, 16 [C07D]

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