ASTEX THERAPEUTICS LTD

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Patent Activity in the Last 10 Years

Technologies

Intl Class Technology Matters Rank in Class
 
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 77178
 
 
 
C07D HETEROCYCLIC COMPOUNDS 63100
 
 
 
A01N PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF 986
 
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 643
 
 
 
C07C ACYCLIC OR CARBOCYCLIC COMPOUNDS 3135
 
 
 
C12N MICRO-ORGANISMS OR ENZYMES; COMPOSITIONS THEREOF 2165
 
 
 
G01N INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES 2204
 
 
 
C04B LIME; MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS 167
 
 
 
C07F ACYCLIC, CARBOCYCLIC, OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM, OR TELLURIUM 169
 
 
 
C12Q MEASURING OR TESTING PROCESSES INVOLVING ENZYMES OR MICRO-ORGANISMS 1124

Top Patents (by citation)

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Recent Publications

Publication # Title Filing Date Pub Date Intl Class
2018/0065,959 BICYCLIC HETEROCYCLE COMPOUNDS AND THEIR USES IN THERAPYAug 11, 17Mar 08, 18[A61K, C07D]
2018/0021,332 PHARMACEUTICAL COMPOSITIONS COMPRISING N-(3,5-DIMETHOXYPHENYL)-N'-(1-METHYLETHYL)-N-[3-(1-METHYL-1H-PYRAZOL-4-YL)QUINOXALIN-6-YL]ETHANE-1,2-DIAMINEFeb 09, 16Jan 25, 18[A61K]
2017/0334,907 BICYCLIC HETEROCYCLE COMPOUNDS AND THEIR USES IN THERAPYMay 03, 17Nov 23, 17[A61K, C07D]
2017/0100,406 COMBINATIONS OF AN FGFR INHIBITOR AND AN IGF1R INHIBITORMar 26, 15Apr 13, 17[A61K]
2016/0311,800 PYRAZOLYL QUINOXALINE KINASE INHIBITORSApr 28, 16Oct 27, 16[C07F, C07D]
2016/0039,832 SALT(S) OF 7-CYCLOPENTYL-2-(5-PIPERAZIN-1-YL-PYRIDIN-2-YLAMINO)-7H-PYRROLO[2,3-D]PYRIMIDINE-6-CARBOXYLIC ACID DIMETHYLAMIDE AND PROCESSES OF MAKING THEREOFOct 20, 15Feb 11, 16[C07D, C07C]
2016/0031,856 SUBSTITUTED QUINOXALINES AS FGFR KINASE INHIBITORSAug 03, 15Feb 04, 16[C07D]

Recent Patents

Patent # Title Filing Date Issue Date Intl Class
9914719 Hydroxybenzamide derivatives and their use as inhibitors of HSP90Aug 25, 14Mar 13, 18[A61K, C07D, C07C]
9902714 Quinoxaline derivatives useful as FGFR kinase modulatorsMar 26, 15Feb 27, 18[A61K, C07D, A61P]
9856236 Substituted quinoxalines as FGFR kinase inhibitorsAug 03, 15Jan 02, 18[C07D]
9850228 Pyrazolyl quinoxaline kinase inhibitorsApr 28, 16Dec 26, 17[A61K, C07F, C07D]
9783538 Bicyclic heterocycle compounds and their uses in therapyDec 19, 14Oct 10, 17[A61K, C07D]
9757364 Naphthyridine derivative compoundsOct 31, 16Sep 12, 17[A61K]
9737544 CompoundsJan 19, 16Aug 22, 17[A61K, C07D]
9730912 Pharmaceutical compoundsOct 12, 07Aug 15, 17[A61K]
9676768 Bicyclic heterocycle compounds and their uses in therapyMar 20, 15Jun 13, 17[A61K, C07D]
9663512 Bicyclic heterocycle compounds and their uses in therapyOct 18, 13May 30, 17[C07D]

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Expired/Abandoned/Withdrawn Patents

Patent # Title Status Filing Date Issue/Pub Date Intl Class
2017/0183,352 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USESAbandonedAug 08, 16Jun 29, 17[A61K, C07D]
9145394 Substituted quinoxalines as FGFR kinase inhibitorsWithdrawnNov 29, 11Sep 29, 15[A61K, C07D]
2014/0288,040 SUBSTITUTED BENZYLAMINE COMPOUNDS, THEIR USE IN MEDICINE, AND IN PARTICULAR THE TREATMENT OF HEPATITIS C VIRUS (HCV) INFECTIONAbandonedOct 31, 12Sep 25, 14[A61K, C07D, C07C]
2014/0010,892 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORSAbandonedMay 24, 13Jan 09, 14[A61K, C07D]
8598217 Imidazole derivatives and their use as modulators of cyclin dependent kinasesExpiredApr 30, 10Dec 03, 13[A61K, C07D, A61P]
8541461 Pharmaceutical combinations comprising pyrazole derivatives as protein kinase modulatorsExpiredJun 21, 06Sep 24, 13[A61K]
8435970 Pharmaceutical combinations of 1-cyclopropyl-3-[3-(5-morpholin-4-ylmethyl-1H-benzoimidazol-2-yl)-1H-pyrazol-4-yl]-ureaExpiredJun 29, 07May 07, 13[A61K]
8399442 Pharmaceutical compoundsExpiredDec 29, 06Mar 19, 13[A61K]
8367687 Pyrazole derivativesExpiredDec 08, 08Feb 05, 13[A61K, A01N]
2012/0207,763 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USESAbandonedApr 20, 12Aug 16, 12[A61K, A61P]
8110573 Pyrazole compounds that modulate the activity of CDK, GSK and aurora kinasesExpiredDec 30, 05Feb 07, 12[A61K, C07D]
2011/0224,203 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORSAbandonedMay 26, 11Sep 15, 11[A61K, A61P]
7977477 Benzimidazole derivatives and their use as protein kinase inhibitorsExpiredJul 05, 04Jul 12, 11[A61K, C07D]
2011/0159,111 PHARMACEUTICAL COMBINATIONSAbandonedJun 29, 07Jun 30, 11[A61K, A61P]
7951819 Imidazo[4, 5-B]pyridin-2-one and oxazolo[4, 5-B] pyridin-2-one compounds and analogs thereof as cancer therapeutic compoundsExpiredApr 26, 07May 31, 11[A61K, A01N, C07D]
2010/0324,072 PYRROLOPYRIDINE DERIVATIVES AND THEIR USE AS BACE INHIBITORSAbandonedMay 14, 08Dec 23, 10[A61K, C07D, A61P]
2010/0298,340 Thiazol-Guanidine Derivatives Useful As A (Beta)-Related PathologiesAbandonedApr 12, 07Nov 25, 10[A61K, C07D, C12N, C07C, A61P]
2010/0210,617 Aryl-Alkylamines And Heteroaryl-Alkylamines As Protein Kinase InhibitorsAbandonedJun 21, 06Aug 19, 10[A61K, C07D, A61P]
2010/0160,324 PYRAZOLE DERIVATIVES AS THAT MODULATE THE ACTIVITY OF CDK, GSK AND AURORA KINASESAbandonedDec 30, 05Jun 24, 10[A61K, C07D, A61P]
2010/0120,798 SUBSTITUTED PIPERIDINES CONTAINING A HETEROARYLAMIDE OR HETEROARYLPHENYL MOIETYAbandonedDec 20, 07May 13, 10[A61K, C07D, A61P]

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